Cole, Derek C

Conformationally constrained N1-arylsulfonyltryptamine derivatives as 5-HT6 receptor antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Nov 2005 - 4780-5 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2005.07.028 doi


Adenylyl Cyclases--metabolism
Cyclic AMP--biosynthesis
Humans
Molecular Conformation
Protein Binding
Receptors, Serotonin--drug effects
Serotonin Antagonists--chemical synthesis
Serotonin Receptor Agonists--chemical synthesis
Structure-Activity Relationship
Tryptamines--chemical synthesis