Brautigan, D L

Allosteric activation of protein phosphatase 2C by D-chiro-inositol-galactosamine, a putative mediator mimetic of insulin action. [electronic resource] - Biochemistry Aug 2005 - 11067-73 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.

0006-2960

10.1021/bi0508845 doi


Amino Acid Substitution--genetics
Animals
Binding Sites--genetics
Blood Glucose--drug effects
Chelating Agents--administration & dosage
Diabetes Mellitus, Experimental--drug therapy
Dose-Response Relationship, Drug
Drug Synergism
Enzyme Activation--drug effects
Galactosamine--administration & dosage
Hydrogen Bonding--drug effects
Inositol--administration & dosage
Inositol Phosphates--administration & dosage
Insulin--administration & dosage
Male
Manganese--chemistry
Models, Molecular
Nitrophenols--chemistry
Organophosphorus Compounds--chemistry
Phosphoprotein Phosphatases--chemistry
Point Mutation
Protein Binding--genetics
Protein Phosphatase 2C
Protein Structure, Tertiary--genetics
Rats
Rats, Sprague-Dawley