Wolff, Christian
[3H]linopirdine binding to rat brain membranes is not relevant for M-channel interaction. [electronic resource]
- European journal of pharmacology Jul 2005
- 10-7 p. digital
Publication Type: Comparative Study; Journal Article
ISSN: 0014-2999
Standard No.: 10.1016/j.ejphar.2005.06.005 doi
Subjects--Topical Terms: Animals Anthracenes--pharmacology Binding, Competitive--drug effects Brain--metabolism CHO Cells Cell Membrane--metabolism Chlorides--metabolism Cricetinae Cricetulus Cytochrome P-450 CYP2D6--metabolism Cytochrome P-450 CYP3A Cytochrome P-450 Enzyme System--metabolism Dose-Response Relationship, Drug Indoles--metabolism KCNQ3 Potassium Channel Ketoconazole--pharmacology Kinetics Liver--metabolism Male Miconazole--pharmacology Potassium Channels, Voltage-Gated--antagonists & inhibitors Pyridines--metabolism Pyrilamine--pharmacology Quinidine--pharmacology Radioligand Assay Rats Rats, Sprague-Dawley Rubidium--metabolism Tritium