Wolff, Christian

[3H]linopirdine binding to rat brain membranes is not relevant for M-channel interaction. [electronic resource] - European journal of pharmacology Jul 2005 - 10-7 p. digital

Publication Type: Comparative Study; Journal Article

0014-2999

10.1016/j.ejphar.2005.06.005 doi


Animals
Anthracenes--pharmacology
Binding, Competitive--drug effects
Brain--metabolism
CHO Cells
Cell Membrane--metabolism
Chlorides--metabolism
Cricetinae
Cricetulus
Cytochrome P-450 CYP2D6--metabolism
Cytochrome P-450 CYP3A
Cytochrome P-450 Enzyme System--metabolism
Dose-Response Relationship, Drug
Indoles--metabolism
KCNQ3 Potassium Channel
Ketoconazole--pharmacology
Kinetics
Liver--metabolism
Male
Miconazole--pharmacology
Potassium Channels, Voltage-Gated--antagonists & inhibitors
Pyridines--metabolism
Pyrilamine--pharmacology
Quinidine--pharmacology
Radioligand Assay
Rats
Rats, Sprague-Dawley
Rubidium--metabolism
Tritium