Matasi, Julius J

2-(2-Furanyl)-7-phenyl[1,2,4]triazolo[1,5-c]pyrimidin-5-amine analogs as adenosine A2A antagonists: the successful reduction of hERG activity. Part 2. [electronic resource] - Bioorganic & medicinal chemistry letters Aug 2005 - 3675-8 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2005.05.043 doi


Adenosine A2 Receptor Antagonists
Administration, Oral
Animals
Catalepsy--drug therapy
Disease Models, Animal
Drug Evaluation, Preclinical
Humans
Molecular Structure
Motor Activity--drug effects
Pyrimidines--chemistry
Rats
Structure-Activity Relationship
Triazoles--chemistry