Barrett, David G P2-P3 conformationally constrained ketoamide-based inhibitors of cathepsin K. [electronic resource] - Bioorganic & medicinal chemistry letters Aug 2005 - 3540-6 p. digital Publication Type: Journal Article ISSN: 0960-894X Standard No.: 10.1016/j.bmcl.2005.05.062 doi Subjects--Topical Terms: Amides--chemical synthesisAnimalsBinding SitesBiological AvailabilityBone Resorption--drug therapyCathepsin KCathepsins--antagonists & inhibitorsCysteine Proteinase Inhibitors--chemical synthesisDisease Models, AnimalHypocalcemia--drug therapyKetones--chemical synthesisRatsRats, WistarSolubilityStructure-Activity Relationship