TY - GEN AU - Burgos-Lepley,Carmen E AU - Thompson,Lisa R AU - Kneen,Clare O AU - Osborne,Simon A AU - Bryans,Justin S AU - Capiris,Thomas AU - Suman-Chauhan,Nirmala AU - Dooley,David J AU - Donovan,Cindy M AU - Field,Mark J AU - Vartanian,Mark G AU - Kinsora,Jack J AU - Lotarski,Susan M AU - El-Kattan,Ayman AU - Walters,Karen AU - Cherukury,Madhu AU - Taylor,Charles P AU - Wustrow,David J AU - Schwarz,Jacob B TI - Carboxylate bioisosteres of gabapentin SN - 0960-894X PY - 2006///0626 KW - Amines KW - chemical synthesis KW - Animals KW - Anticonvulsants KW - Carboxylic Acids KW - chemistry KW - Cyclohexanecarboxylic Acids KW - Disease Models, Animal KW - Dose-Response Relationship, Drug KW - Drug Design KW - Drug Evaluation, Preclinical KW - Gabapentin KW - In Vitro Techniques KW - Mice KW - Mice, Inbred DBA KW - Molecular Structure KW - Rats KW - Stereoisomerism KW - Structure-Activity Relationship KW - Tetrazoles KW - gamma-Aminobutyric Acid N1 - Publication Type: Comparative Study; Journal Article UR - https://doi.org/10.1016/j.bmcl.2005.05.016 ER -