A fluoroquinolone resistance protein from Mycobacterium tuberculosis that mimics DNA. [electronic resource]
- Science (New York, N.Y.) Jun 2005
- 1480-3 p. digital
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.
1095-9203
10.1126/science.1110699 doi
Amino Acid Sequence Antitubercular Agents--chemistry Bacterial Proteins--chemistry Ciprofloxacin--pharmacology Crystallography, X-Ray DNA Gyrase--metabolism DNA, Bacterial--chemistry DNA, Superhelical--chemistry Drug Resistance, Bacterial Drug Resistance, Microbial--physiology Enzyme Inhibitors--chemistry Escherichia coli--enzymology Fluoroquinolones--antagonists & inhibitors Models, Molecular Molecular Mimicry Molecular Sequence Data Monomeric GTP-Binding Proteins Mycobacterium tuberculosis--drug effects Protein Conformation Protein Folding Structure-Activity Relationship Topoisomerase II Inhibitors