Orally administered lenalidomide (CC-5013) is anti-angiogenic in vivo and inhibits endothelial cell migration and Akt phosphorylation in vitro. [electronic resource]
- Microvascular research Jan 2005
- 56-63 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0026-2862
10.1016/j.mvr.2005.01.002 doi
Administration, Oral Angiogenesis Inhibitors--pharmacology Animals Area Under Curve Cell Movement--drug effects Dose-Response Relationship, Drug Endothelium, Vascular--cytology Humans Kinetics Lenalidomide Male Mesentery--blood supply Phosphorylation--drug effects Protein Serine-Threonine Kinases--metabolism Proto-Oncogene Proteins--metabolism Proto-Oncogene Proteins c-akt Rats Rats, Sprague-Dawley Thalidomide--administration & dosage Umbilical Veins--cytology