Benyumov, Alexey O

Anti-proliferative and anti-leukemic activity of DDE46 (compound WHI-07), a novel bromomethoxylated arylphosphate derivative of zidovudine, and related compounds. Studies using human acute lymphoblastic leukemia cells and the zebrafish model. [electronic resource] - Arzneimittel-Forschung 2005 - 114-22 p. digital

Publication Type: Journal Article

0004-4172

10.1055/s-0031-1296832 doi


Animals
Antineoplastic Agents--pharmacology
Apoptosis--drug effects
Caspase Inhibitors
Cell Proliferation--drug effects
Dideoxynucleotides
Drug Screening Assays, Antitumor
Humans
Jurkat Cells
Leukemia--drug therapy
Magnetic Resonance Spectroscopy
Nephelometry and Turbidimetry
Prodrugs--pharmacology
Tetrazolium Salts
Thiazoles
Thymidine Monophosphate--analogs & derivatives
Tubulin--biosynthesis
Zebrafish
Zidovudine--analogs & derivatives