TY - GEN AU - Palmer,Brian D AU - Smaill,Jeff B AU - Rewcastle,Gordon W AU - Dobrusin,Ellen M AU - Kraker,Alan AU - Moore,Charles W AU - Steinkampf,Randall W AU - Denny,William A TI - Structure-activity relationships for 2-anilino-6-phenylpyrido[2,3-d]pyrimidin-7(8H)-ones as inhibitors of the cellular checkpoint kinase Wee1 SN - 0960-894X PY - 2005///0805 KW - Aniline Compounds KW - chemistry KW - CSK Tyrosine-Protein Kinase KW - Cell Cycle Proteins KW - antagonists & inhibitors KW - Cells, Cultured KW - Checkpoint Kinase 1 KW - Enzyme Inhibitors KW - chemical synthesis KW - Humans KW - Inhibitory Concentration 50 KW - Naphthyridines KW - Nuclear Proteins KW - Protein Kinases KW - drug effects KW - Protein-Tyrosine Kinases KW - Pyrimidinones KW - Solubility KW - Structure-Activity Relationship KW - src-Family Kinases N1 - Publication Type: Journal Article UR - https://doi.org/10.1016/j.bmcl.2005.01.079 ER -