Palmer, Brian D

Structure-activity relationships for 2-anilino-6-phenylpyrido[2,3-d]pyrimidin-7(8H)-ones as inhibitors of the cellular checkpoint kinase Wee1. [electronic resource] - Bioorganic & medicinal chemistry letters Apr 2005 - 1931-5 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2005.01.079 doi


Aniline Compounds--chemistry
CSK Tyrosine-Protein Kinase
Cell Cycle Proteins--antagonists & inhibitors
Cells, Cultured
Checkpoint Kinase 1
Enzyme Inhibitors--chemical synthesis
Humans
Inhibitory Concentration 50
Naphthyridines--chemistry
Nuclear Proteins--antagonists & inhibitors
Protein Kinases--drug effects
Protein-Tyrosine Kinases--antagonists & inhibitors
Pyrimidinones--chemistry
Solubility
Structure-Activity Relationship
src-Family Kinases