Ojima, Iwao

Design, synthesis and structure-activity relationships of novel taxane-based multidrug resistance reversal agents. [electronic resource] - Journal of medicinal chemistry Mar 2005 - 2218-28 p. digital

Publication Type: Journal Article; Research Support, U.S. Gov't, P.H.S.

0022-2623

10.1021/jm049483y doi


ATP Binding Cassette Transporter, Subfamily B, Member 1--metabolism
Antineoplastic Agents--chemical synthesis
Cell Line, Tumor
Combinatorial Chemistry Techniques
Drug Resistance, Multiple--drug effects
Drug Resistance, Neoplasm--drug effects
Drug Screening Assays, Antitumor
Humans
Hydrophobic and Hydrophilic Interactions
Mitoxantrone--metabolism
Multidrug Resistance-Associated Proteins--metabolism
Paclitaxel--pharmacology
Structure-Activity Relationship
Taxoids--chemical synthesis