Design and optimization of tricyclic phtalimide analogues as novel inhibitors of HIV-1 integrase. [electronic resource]
- Journal of medicinal chemistry Mar 2005
- 1930-40 p. digital
Publication Type: Journal Article
0022-2623
10.1021/jm049559q doi
Anti-HIV Agents--chemical synthesis Binding Sites Cell Line HIV Integrase--chemistry HIV Integrase Inhibitors--chemical synthesis HIV-1--drug effects Heterocyclic Compounds, 3-Ring--chemical synthesis Humans Models, Molecular Phthalimides--chemical synthesis Protein Binding Pyrroles--chemical synthesis Quinoxalines--chemical synthesis Structure-Activity Relationship