Rational design, synthesis, and structure-activity relationships of aryltriazoles as novel corticotropin-releasing factor-1 receptor antagonists. [electronic resource]
- Journal of medicinal chemistry Mar 2005
- 1540-9 p. digital
Publication Type: Journal Article
0022-2623
10.1021/jm049339c doi
Animals Blood-Brain Barrier--metabolism Cell Line Cyclic AMP--biosynthesis Drug Design Fibroblasts--metabolism Humans Male Mice Models, Molecular Molecular Conformation Radioligand Assay Rats Rats, Sprague-Dawley Receptors, Corticotropin-Releasing Hormone--antagonists & inhibitors Stereoisomerism Structure-Activity Relationship Triazoles--chemical synthesis CRF Receptor, Type 1