Lowe, Richard F

Rational design, synthesis, and structure-activity relationships of aryltriazoles as novel corticotropin-releasing factor-1 receptor antagonists. [electronic resource] - Journal of medicinal chemistry Mar 2005 - 1540-9 p. digital

Publication Type: Journal Article

0022-2623

10.1021/jm049339c doi


Animals
Blood-Brain Barrier--metabolism
Cell Line
Cyclic AMP--biosynthesis
Drug Design
Fibroblasts--metabolism
Humans
Male
Mice
Models, Molecular
Molecular Conformation
Radioligand Assay
Rats
Rats, Sprague-Dawley
Receptors, Corticotropin-Releasing Hormone--antagonists & inhibitors
Stereoisomerism
Structure-Activity Relationship
Triazoles--chemical synthesis
CRF Receptor, Type 1