Do drug substrates enter the common drug-binding pocket of P-glycoprotein through "gates"? [electronic resource]
- Biochemical and biophysical research communications Apr 2005
- 419-22 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0006-291X
10.1016/j.bbrc.2005.01.134 doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--chemistry Animals Binding Sites Drug Resistance--physiology Humans Ion Channel Gating--physiology Models, Biological Models, Chemical Pharmaceutical Preparations--chemistry Protein Binding Protein Conformation Structure-Activity Relationship