Doss, George A Metabolic activation of a 1,3-disubstituted piperazine derivative: evidence for a novel ring contraction to an imidazoline. [electronic resource] - Chemical research in toxicology Feb 2005 - 271-6 p. digital Publication Type: Journal Article ISSN: 0893-228X Standard No.: 10.1021/tx049711r doi Subjects--Topical Terms: AnimalsBile--drug effectsBiotransformationCyclizationGlutathione--drug effectsHumansImidazolines--chemical synthesisMaleMicrosomes, Liver--drug effectsMolecular StructureNADP--drug effectsPiperazines--administration & dosageProtein BindingRatsRats, Sprague-Dawley