TY - GEN AU - Wu,Wen-Lian AU - Burnett,Duane A AU - Spring,Richard AU - Greenlee,William J AU - Smith,Michelle AU - Favreau,Leonard AU - Fawzi,Ahmad AU - Zhang,Hongtao AU - Lachowicz,Jean E TI - Dopamine D1/D5 receptor antagonists with improved pharmacokinetics: design, synthesis, and biological evaluation of phenol bioisosteric analogues of benzazepine D1/D5 antagonists SN - 0022-2623 PY - 2005///0307 KW - Animals KW - Benzazepines KW - chemical synthesis KW - Cell Line KW - Cricetinae KW - Cricetulus KW - Cyclic AMP KW - biosynthesis KW - Dopamine Antagonists KW - Drug Design KW - Male KW - Models, Molecular KW - Phenols KW - Radioligand Assay KW - Rats KW - Rats, Sprague-Dawley KW - Receptors, Dopamine D1 KW - antagonists & inhibitors KW - Receptors, Dopamine D5 KW - Structure-Activity Relationship N1 - Publication Type: Journal Article UR - https://doi.org/10.1021/jm030614p ER -