Wu, Wen-Lian

Dopamine D1/D5 receptor antagonists with improved pharmacokinetics: design, synthesis, and biological evaluation of phenol bioisosteric analogues of benzazepine D1/D5 antagonists. [electronic resource] - Journal of medicinal chemistry Feb 2005 - 680-93 p. digital

Publication Type: Journal Article

0022-2623

10.1021/jm030614p doi


Animals
Benzazepines--chemical synthesis
Cell Line
Cricetinae
Cricetulus
Cyclic AMP--biosynthesis
Dopamine Antagonists--chemical synthesis
Drug Design
Male
Models, Molecular
Phenols--chemical synthesis
Radioligand Assay
Rats
Rats, Sprague-Dawley
Receptors, Dopamine D1--antagonists & inhibitors
Receptors, Dopamine D5
Structure-Activity Relationship