Trifilieff, Alexandre

CGH2466, a combined adenosine receptor antagonist, p38 mitogen-activated protein kinase and phosphodiesterase type 4 inhibitor with potent in vitro and in vivo anti-inflammatory activities. [electronic resource] - British journal of pharmacology Apr 2005 - 1002-10 p. digital

Publication Type: Comparative Study; Journal Article

0007-1188

10.1038/sj.bjp.0706132 doi


3',5'-Cyclic-AMP Phosphodiesterases--antagonists & inhibitors
Animals
Anti-Inflammatory Agents, Non-Steroidal--chemistry
Cricetinae
Cyclic Nucleotide Phosphodiesterases, Type 3
Cyclic Nucleotide Phosphodiesterases, Type 4
Dose-Response Relationship, Drug
Female
Humans
Imidazoles--chemistry
Mice
Mice, Inbred BALB C
Mice, Inbred C57BL
Phosphodiesterase Inhibitors--chemistry
Protein Kinase Inhibitors--chemistry
Purinergic P1 Receptor Antagonists
Pyridines--chemistry
Receptors, Purinergic P1--metabolism
Thiazoles--chemistry
p38 Mitogen-Activated Protein Kinases--antagonists & inhibitors