Tseng, Ping-Hui

Synergistic interactions between imatinib mesylate and the novel phosphoinositide-dependent kinase-1 inhibitor OSU-03012 in overcoming imatinib mesylate resistance. [electronic resource] - Blood May 2005 - 4021-7 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, Non-P.H.S.; Research Support, U.S. Gov't, P.H.S.

0006-4971

10.1182/blood-2004-07-2967 doi


3-Phosphoinositide-Dependent Protein Kinases
Animals
Antineoplastic Agents--pharmacology
Apoptosis--drug effects
Benzamides
Cell Line, Tumor
Drug Resistance, Neoplasm--drug effects
Drug Synergism
Enzyme Activation--drug effects
Fusion Proteins, bcr-abl--genetics
Imatinib Mesylate
Mice
Mutation--genetics
Phosphorylation
Piperazines--pharmacology
Protein Kinase Inhibitors--pharmacology
Protein Serine-Threonine Kinases--antagonists & inhibitors
Proto-Oncogene Proteins--antagonists & inhibitors
Proto-Oncogene Proteins c-akt
Pyrazoles--pharmacology
Pyrimidines--pharmacology
Signal Transduction--drug effects
Sulfonamides--pharmacology