Synthesis and SAR of 5,6-diarylpyridines as human CB1 inverse agonists. [electronic resource]
- Bioorganic & medicinal chemistry letters Feb 2005
- 645-51 p. digital
Publication Type: Journal Article
0960-894X
10.1016/j.bmcl.2004.11.031 doi
Animals Biological Availability CHO Cells Cricetinae Humans Inhibitory Concentration 50 Male Pyridines--chemical synthesis Radioligand Assay Rats Rats, Sprague-Dawley Receptor, Cannabinoid, CB1--agonists Structure-Activity Relationship Tissue Distribution Transfection