TY  - GEN
AU  - Doherty,Elizabeth M
AU  - Fotsch,Christopher
AU  - Bo,Yunxin
AU  - Chakrabarti,Partha P
AU  - Chen,Ning
AU  - Gavva,Narender
AU  - Han,Nianhe
AU  - Kelly,Michael G
AU  - Kincaid,John
AU  - Klionsky,Lana
AU  - Liu,Qingyian
AU  - Ognyanov,Vassil I
AU  - Tamir,Rami
AU  - Wang,Xianghong
AU  - Zhu,Jiawang
AU  - Norman,Mark H
AU  - Treanor,James J S
TI  - Discovery of potent, orally available vanilloid receptor-1 antagonists. Structure-activity relationship of N-aryl cinnamides
SN  - 0022-2623
PY  - 2005///0217
KW  - Administration, Oral
KW  - Animals
KW  - Biochemistry
KW  - methods
KW  - Biological Availability
KW  - CHO Cells
KW  - drug effects
KW  - Calcium
KW  - metabolism
KW  - Capsaicin
KW  - pharmacology
KW  - Cinnamates
KW  - chemistry
KW  - Cricetinae
KW  - Cricetulus
KW  - Humans
KW  - Hydrogen-Ion Concentration
KW  - Inhibitory Concentration 50
KW  - Ion Channels
KW  - antagonists & inhibitors
KW  - Male
KW  - Rats
KW  - Rats, Sprague-Dawley
KW  - Recombinant Proteins
KW  - Structure-Activity Relationship
KW  - TRPV Cation Channels
N1  - Publication Type: Journal Article
UR  - https://doi.org/10.1021/jm049485i
ER  -