Doherty, Elizabeth M <br/><br/>
Discovery of potent, orally available vanilloid receptor-1 antagonists. Structure-activity relationship of N-aryl cinnamides.  [electronic resource] 

 -  Journal of medicinal chemistry  Jan 2005 
 - 71-90 p.  digital 
<br/><br/> Publication Type: Journal Article 
<br/><br/><label>ISSN: </label>0022-2623 
<br/><br/><label>Standard No.: </label>10.1021/jm049485i  doi 
<br/><br/><label>Subjects--Topical Terms: </label><br/>Administration, Oral<br/>Animals<br/>Biochemistry--methods<br/>Biological Availability<br/>CHO Cells--drug effects<br/>Calcium--metabolism<br/>Capsaicin--pharmacology<br/>Cinnamates--chemistry<br/>Cricetinae<br/>Cricetulus<br/>Humans<br/>Hydrogen-Ion Concentration<br/>Inhibitory Concentration 50<br/>Ion Channels--antagonists & inhibitors<br/>Male<br/>Rats<br/>Rats, Sprague-Dawley<br/>Recombinant Proteins--drug effects<br/>Structure-Activity Relationship<br/>TRPV Cation Channels