Cole, Derek C

N1-arylsulfonyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole derivatives are potent and selective 5-HT6 receptor antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Jan 2005 - 379-83 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2004.10.064 doi


Adenylyl Cyclases--metabolism
HeLa Cells
Humans
Indoles--chemical synthesis
Receptors, Serotonin--metabolism
Serotonin Antagonists--chemical synthesis
Structure-Activity Relationship