Cole, Derek C N1-arylsulfonyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole derivatives are potent and selective 5-HT6 receptor antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Jan 2005 - 379-83 p. digital Publication Type: Journal Article ISSN: 0960-894X Standard No.: 10.1016/j.bmcl.2004.10.064 doi Subjects--Topical Terms: Adenylyl Cyclases--metabolismHeLa CellsHumansIndoles--chemical synthesisReceptors, Serotonin--metabolismSerotonin Antagonists--chemical synthesisStructure-Activity Relationship