Salvati, Mark E

Structure based approach to the design of bicyclic-1H-isoindole-1,3(2H)-dione based androgen receptor antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Jan 2005 - 271-6 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2004.10.085 doi


Androgen Antagonists--chemical synthesis
Bridged Bicyclo Compounds, Heterocyclic--chemical synthesis
Indoles--chemistry
Protein Isoforms
Receptors, Androgen--metabolism
Structure-Activity Relationship
Tumor Cells, Cultured