Ferrari, Flora
Pharmacological profile of CR3465, a new leukotriene CysLT1 receptor antagonist with broad anti-inflammatory activity. [electronic resource]
- European journal of pharmacology Nov 2004
- 223-33 p. digital
Publication Type: Journal Article
ISSN: 0014-2999
Standard No.: 10.1016/j.ejphar.2004.10.010 doi
Subjects--Topical Terms: 3',5'-Cyclic-AMP Phosphodiesterases--antagonists & inhibitors Animals Anti-Inflammatory Agents Bronchoalveolar Lavage Fluid--cytology Bronchoconstriction--drug effects Cell Degranulation--drug effects Cyclic Nucleotide Phosphodiesterases, Type 3 Cyclic Nucleotide Phosphodiesterases, Type 4 Guinea Pigs Histamine--pharmacology Histamine Antagonists--pharmacology Humans In Vitro Techniques Leukotriene D4--antagonists & inhibitors Membrane Proteins--antagonists & inhibitors N-Formylmethionine Leucyl-Phenylalanine--pharmacology Neutrophils--drug effects Parasympatholytics--pharmacology Peroxidase--metabolism Phosphodiesterase Inhibitors--pharmacology Quinolines--pharmacology Radioligand Assay Rats Receptors, Leukotriene Tumor Necrosis Factor-alpha--metabolism Tyrosine--analogs & derivatives