Chambers, Mark S

An orally bioavailable, functionally selective inverse agonist at the benzodiazepine site of GABAA alpha5 receptors with cognition enhancing properties. [electronic resource] - Journal of medicinal chemistry Nov 2004 - 5829-32 p. digital

Publication Type: Journal Article

0022-2623

10.1021/jm040863t doi


Administration, Oral
Animals
Binding Sites
Biological Availability
Cognition--drug effects
Dogs
GABA-A Receptor Agonists
Isoxazoles--adverse effects
Maze Learning--drug effects
Mice
Nootropic Agents--adverse effects
Patch-Clamp Techniques
Protein Subunits
Radioligand Assay
Rats
Receptors, GABA-A--metabolism
Triazines--adverse effects