Chambers, Mark S An orally bioavailable, functionally selective inverse agonist at the benzodiazepine site of GABAA alpha5 receptors with cognition enhancing properties. [electronic resource] - Journal of medicinal chemistry Nov 2004 - 5829-32 p. digital Publication Type: Journal Article ISSN: 0022-2623 Standard No.: 10.1021/jm040863t doi Subjects--Topical Terms: Administration, OralAnimalsBinding SitesBiological AvailabilityCognition--drug effectsDogsGABA-A Receptor AgonistsIsoxazoles--adverse effectsMaze Learning--drug effectsMiceNootropic Agents--adverse effectsPatch-Clamp TechniquesProtein SubunitsRadioligand AssayRatsReceptors, GABA-A--metabolismTriazines--adverse effects