Deutsch, E

Tyrosine kinase inhibitor AG1024 exerts antileukaemic effects on STI571-resistant Bcr-Abl expressing cells and decreases AKT phosphorylation. [electronic resource] - British journal of cancer Nov 2004 - 1735-41 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

0007-0920

10.1038/sj.bjc.6602190 doi


Animals
Antineoplastic Agents--therapeutic use
Benzamides
Cell Proliferation--drug effects
DNA-Activated Protein Kinase
DNA-Binding Proteins--antagonists & inhibitors
Drug Resistance, Neoplasm
Enzyme Inhibitors--therapeutic use
Fusion Proteins, bcr-abl
Gene Expression Regulation, Leukemic
Humans
Imatinib Mesylate
Leukemia, Erythroblastic, Acute--drug therapy
Mice
Mice, Nude
Neoplasm Recurrence, Local--drug therapy
Nuclear Proteins
Phosphorylation
Piperazines--pharmacology
Protein Serine-Threonine Kinases--antagonists & inhibitors
Protein-Tyrosine Kinases--antagonists & inhibitors
Proto-Oncogene Proteins--metabolism
Proto-Oncogene Proteins c-akt
Pyrimidines--pharmacology
Tumor Cells, Cultured
Tyrphostins--therapeutic use