Inhibition of Chk1 by the G2 DNA damage checkpoint inhibitor isogranulatimide. [electronic resource]
- Molecular cancer therapeutics Oct 2004
- 1221-7 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
1535-7163
Antineoplastic Agents--pharmacology Catalytic Domain Cell Line, Tumor Checkpoint Kinase 1 Crystallography, X-Ray Cysteine--chemistry DNA Damage Dose-Response Relationship, Drug G2 Phase Glutamine--chemistry Glycogen Synthase Kinase 3--metabolism Glycogen Synthase Kinase 3 beta Humans Imidazoles--pharmacology Indoles--antagonists & inhibitors Inhibitory Concentration 50 Maleimides--antagonists & inhibitors Models, Chemical Models, Molecular Nitrogen--chemistry Phenotype Protein Binding Protein Kinase C--metabolism Protein Kinase C beta Protein Kinases--metabolism Protein Structure, Tertiary Time Factors