Lin, Nan-Horng

Synthesis and biological evaluation of 1-benzyl-5-(3-biphenyl-2-yl-propyl)-1H-imidazole as novel farnesyltransferase inhibitor. [electronic resource] - Bioorganic & medicinal chemistry letters Oct 2004 - 5057-62 p. digital

Publication Type: Comparative Study; Journal Article

0960-894X

10.1016/j.bmcl.2004.07.083 doi


Alkyl and Aryl Transferases--antagonists & inhibitors
Animals
Antineoplastic Agents--chemical synthesis
Biological Availability
Biphenyl Compounds--chemical synthesis
Farnesyltranstransferase
Imidazoles--chemical synthesis
In Vitro Techniques
Rats
Structure-Activity Relationship