Investigation of the effect of the farnesyl protein transferase inhibitor R115777 on isoprenylation and intracellular signalling by the prostacyclin receptor. [electronic resource]
- British journal of pharmacology Sep 2004
- 318-30 p. digital
Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
0007-1188
10.1038/sj.bjp.0705956 doi
Alkyl and Aryl Transferases--antagonists & inhibitors Animals Calcium--metabolism Cell Line Cell Survival--drug effects Cyclic AMP--metabolism Dose-Response Relationship, Drug Drug Evaluation, Preclinical--methods Enzyme Inhibitors--pharmacology Humans Iloprost--pharmacology Ireland Mice Molecular Chaperones--drug effects Organophosphonates Protein Prenylation--drug effects Quinolones--chemistry Receptor Cross-Talk--drug effects Receptors, Prostaglandin--classification Time Factors Transfection--methods Transferases--antagonists & inhibitors Tritium