Influence of hepatic and intestinal cytochrome P4503A activity on the acute disposition and effects of oral transmucosal fentanyl citrate. [electronic resource]
- Anesthesiology Sep 2004
- 729-37 p. digital
Publication Type: Clinical Trial; Journal Article; Randomized Controlled Trial; Research Support, U.S. Gov't, P.H.S.
0003-3022
10.1097/00000542-200409000-00022 doi
Adult Analgesics, Opioid--administration & dosage Antibiotics, Antitubercular--pharmacology Antiemetics--pharmacology Area Under Curve Aryl Hydrocarbon Hydroxylases--metabolism Beverages Chromatography, High Pressure Liquid Citrus Cross-Over Studies Cytochrome P-450 CYP3A Drug Interactions Female Fentanyl--administration & dosage Food-Drug Interactions Half-Life Humans Intestines--enzymology Liver--enzymology Male Oxidoreductases, N-Demethylating--metabolism Pupil--drug effects Rifampin--pharmacology Spectrometry, Mass, Electrospray Ionization Troleandomycin--pharmacology