TY - GEN AU - Laufersweiler,Matthew J AU - Brugel,Todd A AU - Clark,Michael P AU - Golebiowski,Adam AU - Bookland,Roger G AU - Laughlin,Steven K AU - Sabat,Mark P AU - Townes,Jennifer A AU - VanRens,John C AU - De,Biswanath AU - Hsieh,Lily C AU - Heitmeyer,Sandra A AU - Juergens,Karen AU - Brown,Kimberly K AU - Mekel,Marlene J AU - Walter,Richard L AU - Janusz,Michael J TI - The development of novel inhibitors of tumor necrosis factor-alpha (TNF-alpha) production based on substituted [5,5]-bicyclic pyrazolones SN - 0960-894X PY - 2005///0223 KW - Administration, Oral KW - Animals KW - Biological Availability KW - Lipopolysaccharides KW - pharmacology KW - Models, Molecular KW - Pyrazolones KW - administration & dosage KW - Rats KW - Structure-Activity Relationship KW - Tumor Necrosis Factor-alpha KW - antagonists & inhibitors N1 - Publication Type: Journal Article UR - https://doi.org/10.1016/j.bmcl.2004.06.001 ER -