Akt/protein kinase B signaling inhibitor-2, a selective small molecule inhibitor of Akt signaling with antitumor activity in cancer cells overexpressing Akt. [electronic resource]
- Cancer research Jul 2004
- 4394-9 p. digital
Publication Type: Journal Article; Research Support, U.S. Gov't, Non-P.H.S.; Research Support, U.S. Gov't, P.H.S.
0008-5472
10.1158/0008-5472.CAN-04-0343 doi
Animals Apoptosis--drug effects Cell Division--drug effects Cell Line, Tumor Cyclic AMP-Dependent Protein Kinases--antagonists & inhibitors Enzyme Inhibitors--pharmacology Female Humans Immediate-Early Proteins JNK Mitogen-Activated Protein Kinases MAP Kinase Signaling System--drug effects Mice Mice, Nude Mitogen-Activated Protein Kinases--antagonists & inhibitors NIH 3T3 Cells Nuclear Proteins Nucleosides--pharmacology Protein Kinase C--antagonists & inhibitors Protein Serine-Threonine Kinases--antagonists & inhibitors Proto-Oncogene Proteins--antagonists & inhibitors Proto-Oncogene Proteins c-akt Pyridazines--pharmacology Signal Transduction--drug effects Substrate Specificity Xenograft Model Antitumor Assays p38 Mitogen-Activated Protein Kinases