Tamoxifen resistance by a conformational arrest of the estrogen receptor alpha after PKA activation in breast cancer. [electronic resource]
- Cancer cell Jun 2004
- 597-605 p. digital
Publication Type: Journal Article
1535-6108
10.1016/j.ccr.2004.05.016 doi
Antineoplastic Agents, Hormonal--pharmacology Binding Sites Blotting, Western Breast Neoplasms--enzymology Cell Division Cell Line, Tumor Cyclic AMP-Dependent Protein Kinases--metabolism Down-Regulation Drug Resistance, Neoplasm Enzyme Activation Enzyme Inhibitors--pharmacology Estradiol--analogs & derivatives Estrogen Receptor Modulators--pharmacology Estrogen Receptor alpha Female Fluorescence Resonance Energy Transfer Fulvestrant Humans Luciferases--metabolism Microscopy, Confocal Models, Biological Nucleic Acid Hybridization Oligonucleotide Array Sequence Analysis Phosphorylation Protein Conformation Protein Structure, Tertiary RNA Interference Receptors, Estrogen--chemistry Serine--chemistry Tamoxifen--pharmacology Time Factors Transcriptional Activation Transfection