The novel estrogen 17alpha-20Z-21-[(4-amino)phenyl]-19-norpregna-1,3,5(10),20-tetraene-3,17beta-diol induces apoptosis in prostate cancer cell lines at nanomolar concentrations in vitro. [electronic resource]
- Molecular cancer therapeutics May 2004
- 587-95 p. digital
Publication Type: Journal Article; Research Support, U.S. Gov't, Non-P.H.S.; Research Support, U.S. Gov't, P.H.S.
1535-7163
Apoptosis--drug effects Blotting, Western Bromodeoxyuridine Caspase 3 Caspases--metabolism Cell Cycle--drug effects Cell Line, Tumor Drug Screening Assays, Antitumor Estradiol--analogs & derivatives Estrogen Receptor alpha--metabolism Estrogen Receptor beta--metabolism Flow Cytometry Humans Male Models, Molecular Prostatic Neoplasms--pathology Protein Binding