Tanitame, Akihiko

Design, synthesis and structure-activity relationship studies of novel indazole analogues as DNA gyrase inhibitors with Gram-positive antibacterial activity. [electronic resource] - Bioorganic & medicinal chemistry letters Jun 2004 - 2857-62 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2004.03.044 doi


Anti-Bacterial Agents--chemical synthesis
DNA Topoisomerases--drug effects
Drug Design
Drug Resistance, Multiple
Enterococcus faecalis--drug effects
Enzyme Inhibitors--chemical synthesis
Gram-Positive Bacteria--drug effects
Humans
Imidazoles--chemical synthesis
Inhibitory Concentration 50
Microbial Sensitivity Tests
Staphylococcaceae--drug effects
Structure-Activity Relationship
Topoisomerase II Inhibitors