Design, synthesis and structure-activity relationship studies of novel indazole analogues as DNA gyrase inhibitors with Gram-positive antibacterial activity. [electronic resource]
- Bioorganic & medicinal chemistry letters Jun 2004
- 2857-62 p. digital
Publication Type: Journal Article
0960-894X
10.1016/j.bmcl.2004.03.044 doi
Anti-Bacterial Agents--chemical synthesis DNA Topoisomerases--drug effects Drug Design Drug Resistance, Multiple Enterococcus faecalis--drug effects Enzyme Inhibitors--chemical synthesis Gram-Positive Bacteria--drug effects Humans Imidazoles--chemical synthesis Inhibitory Concentration 50 Microbial Sensitivity Tests Staphylococcaceae--drug effects Structure-Activity Relationship Topoisomerase II Inhibitors