Design, synthesis, and SAR of 2-dialkylamino-4-arylpyrimidines as potent and selective corticotropin-releasing factor(1) (CRF(1)) receptor antagonists. [electronic resource]
- Bioorganic & medicinal chemistry letters May 2004
- 2083-6 p. digital
Publication Type: Journal Article
0960-894X
10.1016/j.bmcl.2004.02.053 doi
Animals CHO Cells Cricetinae Drug Design Pyrimidines--chemical synthesis Rats Receptors, Corticotropin-Releasing Hormone--antagonists & inhibitors Structure-Activity Relationship CRF Receptor, Type 1