Huang, Charles Q

Design, synthesis, and SAR of 2-dialkylamino-4-arylpyrimidines as potent and selective corticotropin-releasing factor(1) (CRF(1)) receptor antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters May 2004 - 2083-6 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2004.02.053 doi


Animals
CHO Cells
Cricetinae
Drug Design
Pyrimidines--chemical synthesis
Rats
Receptors, Corticotropin-Releasing Hormone--antagonists & inhibitors
Structure-Activity Relationship
CRF Receptor, Type 1