Shi, Zhen-Dan

Macrocyclization in the design of non-phosphorus-containing Grb2 SH2 domain-binding ligands. [electronic resource] - Journal of medicinal chemistry Apr 2004 - 2166-9 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.

0022-2623

10.1021/jm030510e doi


Adaptor Proteins, Signal Transducing
Binding Sites
Cell Line, Tumor
Cyclization
Drug Design
Enzyme-Linked Immunosorbent Assay
GRB2 Adaptor Protein
Humans
Ligands
Models, Molecular
Molecular Mimicry
Oligopeptides--chemistry
Peptides, Cyclic--chemical synthesis
Proteins--metabolism
Receptor, ErbB-2--metabolism
src Homology Domains