Andela, Valentine B

The proteosome inhibitor MG132 attenuates retinoic acid receptor trans-activation and enhances trans-repression of nuclear factor kappaB. Potential relevance to chemo-preventive interventions with retinoids. [electronic resource] - Molecular cancer Mar 2004 - 8 p. digital

Publication Type: Journal Article; Research Support, Non-U.S. Gov't

1476-4598

10.1186/1476-4598-3-8 doi


Active Transport, Cell Nucleus--physiology
Cell Line, Tumor
Cell Nucleus--metabolism
DNA, Neoplasm--metabolism
DNA-Binding Proteins--antagonists & inhibitors
Enzyme Activation--physiology
Gene Expression Regulation--physiology
Humans
Leupeptins--pharmacology
Ligands
Macromolecular Substances--antagonists & inhibitors
Matrix Metalloproteinase 9--metabolism
NF-kappa B--genetics
Neoplasm Metastasis--pathology
Neoplasm Proteins
Protein Transport--physiology
Receptors, Retinoic Acid--antagonists & inhibitors
Repressor Proteins--physiology
Retinoids
Tissue Inhibitor of Metalloproteinase-1--metabolism
Transcriptional Activation--drug effects