Balle, Thomas New alpha(1)-adrenoceptor antagonists derived from the antipsychotic sertindole - carbon-11 labelling and pet examination of brain uptake in the cynomolgus monkey. [electronic resource] - Nuclear medicine and biology Apr 2004 - 327-36 p. digital Publication Type: Comparative Study; Evaluation Study; Journal Article ISSN: 0969-8051 Standard No.: 10.1016/j.nucmedbio.2003.08.012 doi Subjects--Topical Terms: ATP Binding Cassette Transporter, Subfamily B, Member 1--deficiencyAdrenergic alpha-1 Receptor AntagonistsAnimalsAntipsychotic Agents--chemistryBrain--diagnostic imagingCaco-2 CellsCarbon Radioisotopes--chemistryCyclosporine--pharmacologyDrug Evaluation, PreclinicalHumansImidazoles--chemistryIndoles--chemistryIsotope Labeling--methodsKineticsMacaca fascicularisMaleMetabolic Clearance RateMicePositron-Emission Tomography--methodsProtein BindingRadiopharmaceuticals--chemical synthesisReceptors, Adrenergic, alpha-1--metabolism