Shi, Bingzhi

Synthesis and biological evaluation of the binding of dopamine D2/D3 receptor agonist, (R,S)-5-hydroxy-2-(N-propyl-N-(5'-(18)F-fluoropentyl)aminotetralin ((18)F-5-OH-FPPAT) in rodents and nonhuman primates. [electronic resource] - Nuclear medicine and biology Apr 2004 - 303-11 p. digital

Publication Type: Comparative Study; Evaluation Study; Journal Article; Research Support, U.S. Gov't, Non-P.H.S.

0969-8051

10.1016/j.nucmedbio.2003.10.004 doi


Animals
Brain--diagnostic imaging
Dopamine D2 Receptor Antagonists
Drug Evaluation, Preclinical
Humans
Isotope Labeling--methods
Kinetics
Macaca mulatta
Male
Metabolic Clearance Rate
Positron-Emission Tomography--methods
Primates
Protein Binding
Radiopharmaceuticals--chemical synthesis
Rats
Rats, Sprague-Dawley
Receptors, Dopamine D2--metabolism
Receptors, Dopamine D3
Rodentia
Species Specificity
Tetrahydronaphthalenes--chemistry
Tissue Distribution