Synthesis and biological evaluation of the binding of dopamine D2/D3 receptor agonist, (R,S)-5-hydroxy-2-(N-propyl-N-(5'-(18)F-fluoropentyl)aminotetralin ((18)F-5-OH-FPPAT) in rodents and nonhuman primates. [electronic resource]
- Nuclear medicine and biology Apr 2004
- 303-11 p. digital
Publication Type: Comparative Study; Evaluation Study; Journal Article; Research Support, U.S. Gov't, Non-P.H.S.
0969-8051
10.1016/j.nucmedbio.2003.10.004 doi
Animals Brain--diagnostic imaging Dopamine D2 Receptor Antagonists Drug Evaluation, Preclinical Humans Isotope Labeling--methods Kinetics Macaca mulatta Male Metabolic Clearance Rate Positron-Emission Tomography--methods Primates Protein Binding Radiopharmaceuticals--chemical synthesis Rats Rats, Sprague-Dawley Receptors, Dopamine D2--metabolism Receptors, Dopamine D3 Rodentia Species Specificity Tetrahydronaphthalenes--chemistry Tissue Distribution