Eisenberger, Mario A

Phase I and clinical pharmacology of a type I and II, 5-alpha-reductase inhibitor (LY320236) in prostate cancer: elevation of estradiol as possible mechanism of action. [electronic resource] - Urology Jan 2004 - 114-9 p. digital

Publication Type: Clinical Trial; Clinical Trial, Phase I; Comparative Study; Journal Article; Research Support, Non-U.S. Gov't

1527-9995

10.1016/j.urology.2003.08.017 doi


5-alpha Reductase Inhibitors
Adenocarcinoma--blood
Androgen Antagonists--administration & dosage
Androstenediols--blood
Benzoquinones--administration & dosage
Biomarkers, Tumor--blood
Chemical and Drug Induced Liver Injury--etiology
Dihydrotestosterone--blood
Disease-Free Survival
Dose-Response Relationship, Drug
Enzyme Inhibitors--administration & dosage
Estradiol--blood
Humans
Isoenzymes--antagonists & inhibitors
Life Tables
Male
Neoplasm Proteins--antagonists & inhibitors
Orchiectomy
Prostate-Specific Antigen--blood
Prostatic Neoplasms--blood
Safety
Substrate Specificity
Testosterone--blood
Treatment Outcome