Progress in pursuit of therapeutic A2A antagonists: the adenosine A2A receptor selective antagonist KW6002: research and development toward a novel nondopaminergic therapy for Parkinson's disease. [electronic resource]
- Neurology Dec 2003
- S97-100 p. digital
Publication Type: Journal Article; Review
1526-632X
10.1212/01.wnl.0000095219.22086.31 doi
Adenosine A2 Receptor Antagonists Animals Antiparkinson Agents--adverse effects Clinical Trials as Topic--statistics & numerical data Corpus Striatum--cytology Disease Models, Animal Drug Evaluation, Preclinical Dyskinesia, Drug-Induced--prevention & control Globus Pallidus--cytology Humans Levodopa--adverse effects Mice Mice, Knockout Motor Activity--drug effects Neurons--drug effects Oxidopamine Parkinson Disease--drug therapy Parkinsonian Disorders--chemically induced Primates Purines--therapeutic use Rats Receptor, Adenosine A2A--metabolism Receptors, Dopamine D2--deficiency gamma-Aminobutyric Acid--metabolism