Kase, Hiroshi

Progress in pursuit of therapeutic A2A antagonists: the adenosine A2A receptor selective antagonist KW6002: research and development toward a novel nondopaminergic therapy for Parkinson's disease. [electronic resource] - Neurology Dec 2003 - S97-100 p. digital

Publication Type: Journal Article; Review

1526-632X

10.1212/01.wnl.0000095219.22086.31 doi


Adenosine A2 Receptor Antagonists
Animals
Antiparkinson Agents--adverse effects
Clinical Trials as Topic--statistics & numerical data
Corpus Striatum--cytology
Disease Models, Animal
Drug Evaluation, Preclinical
Dyskinesia, Drug-Induced--prevention & control
Globus Pallidus--cytology
Humans
Levodopa--adverse effects
Mice
Mice, Knockout
Motor Activity--drug effects
Neurons--drug effects
Oxidopamine
Parkinson Disease--drug therapy
Parkinsonian Disorders--chemically induced
Primates
Purines--therapeutic use
Rats
Receptor, Adenosine A2A--metabolism
Receptors, Dopamine D2--deficiency
gamma-Aminobutyric Acid--metabolism