The influence of the P-glycoprotein inhibitor zosuquidar trihydrochloride (LY335979) on the brain penetration of paclitaxel in mice. [electronic resource]
- Cancer chemotherapy and pharmacology Feb 2004
- 173-8 p. digital
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
0344-5704
10.1007/s00280-003-0720-y doi
ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors Administration, Oral Algorithms Animals Antineoplastic Agents, Phytogenic--pharmacokinetics Area Under Curve Biological Availability Brain--drug effects Dibenzocycloheptenes--pharmacology Female Injections, Intravenous Mice Mice, Knockout Paclitaxel--pharmacokinetics Quinolines--pharmacology Spectrophotometry, Ultraviolet Tissue Distribution