N-desmethylclozapine, an allosteric agonist at muscarinic 1 receptor, potentiates N-methyl-D-aspartate receptor activity. [electronic resource]
- Proceedings of the National Academy of Sciences of the United States of America Nov 2003
- 13674-9 p. digital
Publication Type: Journal Article
0027-8424
10.1073/pnas.1835612100 doi
Allosteric Site Animals Brain--metabolism Cell Line Clozapine--analogs & derivatives Cricetinae DNA, Complementary--metabolism Dose-Response Relationship, Drug Electrophysiology Guanosine 5'-O-(3-Thiotriphosphate)--metabolism Hippocampus--metabolism Humans Inhibitory Concentration 50 Mutagenesis, Site-Directed Neurons--metabolism Protein Binding Rats Receptor, Muscarinic M1--agonists Receptors, N-Methyl-D-Aspartate--metabolism Time Factors