Urbanski, Maud J 2,5-disubstituted 3,4-dihydro-2H-benzo[b][1,4]thiazepines as potent and selective V2 arginine vasopressin receptor antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Nov 2003 - 4031-4 p. digital Publication Type: Journal Article ISSN: 0960-894X Standard No.: 10.1016/j.bmcl.2003.08.051 doi Subjects--Topical Terms: AnimalsAntidiuretic Hormone Receptor AntagonistsAzepines--chemical synthesisBenzamides--chemical synthesisBenzazepines--chemical synthesisDibenzothiazepines--chemical synthesisDiuresis--drug effectsDrug DesignKineticsMalePyrrolesRatsStructure-Activity Relationship