Urbanski, Maud J

2,5-disubstituted 3,4-dihydro-2H-benzo[b][1,4]thiazepines as potent and selective V2 arginine vasopressin receptor antagonists. [electronic resource] - Bioorganic & medicinal chemistry letters Nov 2003 - 4031-4 p. digital

Publication Type: Journal Article

0960-894X

10.1016/j.bmcl.2003.08.051 doi


Animals
Antidiuretic Hormone Receptor Antagonists
Azepines--chemical synthesis
Benzamides--chemical synthesis
Benzazepines--chemical synthesis
Dibenzothiazepines--chemical synthesis
Diuresis--drug effects
Drug Design
Kinetics
Male
Pyrroles
Rats
Structure-Activity Relationship