TY - GEN AU - Yabuki,Masashi AU - Kon-Ya,Yutaka AU - Kataoka,Masaki AU - Shimizudani,Takeshi AU - Akao,Kyoko AU - Ito,Masaki AU - Kanamaru,Hiroshi AU - Nakatsuka,Iwao TI - Pharmacokinetics of a novel N-methyl-D-aspartate receptor antagonist (SM-18400): identification of an N-acetylated metabolite and pre-clinical assessment of N-acetylation polymorphism SN - 0378-7966 PY - 2003///1006 KW - Acetylation KW - Acetyltransferases KW - metabolism KW - Animals KW - Area Under Curve KW - Biotransformation KW - Chromatography, High Pressure Liquid KW - Cytosol KW - Dogs KW - Excitatory Amino Acid Antagonists KW - pharmacokinetics KW - Humans KW - In Vitro Techniques KW - Indicators and Reagents KW - Kinetics KW - Liver KW - Male KW - Polymorphism, Genetic KW - Quinoxalines KW - Rats KW - Rats, Sprague-Dawley KW - Receptors, N-Methyl-D-Aspartate KW - antagonists & inhibitors KW - Spectrometry, Mass, Electrospray Ionization KW - Subcellular Fractions N1 - Publication Type: Journal Article UR - https://doi.org/10.1007/BF03190863 ER -