Pharmacokinetics of a novel N-methyl-D-aspartate receptor antagonist (SM-18400): identification of an N-acetylated metabolite and pre-clinical assessment of N-acetylation polymorphism. [electronic resource]
- European journal of drug metabolism and pharmacokinetics
- 21-9 p. digital
Publication Type: Journal Article
0378-7966
10.1007/BF03190863 doi
Acetylation Acetyltransferases--metabolism Animals Area Under Curve Biotransformation Chromatography, High Pressure Liquid Cytosol--metabolism Dogs Excitatory Amino Acid Antagonists--pharmacokinetics Humans In Vitro Techniques Indicators and Reagents Kinetics Liver--metabolism Male Polymorphism, Genetic Quinoxalines--pharmacokinetics Rats Rats, Sprague-Dawley Receptors, N-Methyl-D-Aspartate--antagonists & inhibitors Spectrometry, Mass, Electrospray Ionization Subcellular Fractions--metabolism