Yabuki, Masashi

Pharmacokinetics of a novel N-methyl-D-aspartate receptor antagonist (SM-18400): identification of an N-acetylated metabolite and pre-clinical assessment of N-acetylation polymorphism. [electronic resource] - European journal of drug metabolism and pharmacokinetics - 21-9 p. digital

Publication Type: Journal Article

0378-7966

10.1007/BF03190863 doi


Acetylation
Acetyltransferases--metabolism
Animals
Area Under Curve
Biotransformation
Chromatography, High Pressure Liquid
Cytosol--metabolism
Dogs
Excitatory Amino Acid Antagonists--pharmacokinetics
Humans
In Vitro Techniques
Indicators and Reagents
Kinetics
Liver--metabolism
Male
Polymorphism, Genetic
Quinoxalines--pharmacokinetics
Rats
Rats, Sprague-Dawley
Receptors, N-Methyl-D-Aspartate--antagonists & inhibitors
Spectrometry, Mass, Electrospray Ionization
Subcellular Fractions--metabolism