Zhang, Han-Cheng

Macrocyclic bisindolylmaleimides as inhibitors of protein kinase C and glycogen synthase kinase-3. [electronic resource] - Bioorganic & medicinal chemistry letters Sep 2003 - 3049-53 p. digital

Publication Type: Journal Article

0960-894X

10.1016/s0960-894x(03)00644-9 doi


Antineoplastic Agents--chemical synthesis
Cell Line
Cyclization
Enzyme Inhibitors--chemical synthesis
Glycogen Synthase Kinase 3--antagonists & inhibitors
Glycogen Synthase Kinase 3 beta
Humans
Indoles--chemical synthesis
Inhibitory Concentration 50
Isoenzymes--chemical synthesis
Maleimides--chemical synthesis
Protein Kinase C--antagonists & inhibitors
Protein Kinase C beta
Structure-Activity Relationship